http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1724269-A1

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filingDate 2005-05-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1faa49e5bc5c404c27329e6594dd957f
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_56b4d5e132c18cf8fa0a9b4b760f371a
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publicationDate 2006-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1724269-A1
titleOfInvention Heteroaryl-carboxylic acid (sulfamoyl alkyl) amide - derivatives as factor Xa inhibitors
abstract The present invention relates to compounds of the formula I,n nin which R1; R2; R3; V; G1 and G2 have the meanings indicated in the claims. The compounds of the formula I are valuable pharmacologically active compounds. They exhibit a strong antithrombotic effect and are suitable, for example, for the therapy and prophylaxis of cardiovascular disorders like thromboembolic diseases or restenoses. They are reversible inhibitors of the blood clotting enzymes factor Xa, and can in general be applied in conditions in which an undesired activity of factor Xa is present or for the cure or prevention of which an inhibition of factor Xa is intended. The invention furthermore relates to processes for the preparation of compounds of the formula I, their use, in particular as active ingredients in pharmaceuticals, and pharmaceutical preparations comprising them.
priorityDate 2005-05-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 492.