http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1720903-A1

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filingDate 2005-01-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ca1e925e48651e52b133fc2cc70bbcfc
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1c8e7e71f15f76c87d5d45359942c099
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_12db1e8d469dfe4867bcb9ea3a1d7a74
publicationDate 2006-11-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1720903-A1
titleOfInvention Corticotropin-releasing factor receptor 1 (crfr1) agonist polypeptides
abstract The present invention relates to a compound which is highly selective for CRFR1 without having any significant cross-reactivity for corticotropin-releasing-factor­receptor-2 (CRFR2) and/or corticotropin-releasing-factor-binding protein (CRFBP), said compound comprising or alternatively consisting of the amino acid sequence as depicted in SEQ ID No: 1. In another aspect, the present invention relates to a pharmaceutical and/or diagnostic composition comprising the novel CRFR1 agonist of the present invention. The present invention also provides a kit comprising the novel CRFR1 agonist of the present invention and optionally instructions to use. Furthermore, the present invention provides the use of the compound of the present invention for the preparation of a pharmaceutical composition for the treatment of depression and, additionally, the use of the compound of the present invention for the preparation of a diagnostic composition for the determination of pituitary corticotroph responsiveness and/or for differentiating pituitary and ectopic production of ACTH in patients with ACTH-dependent Cushing's syndrome.
priorityDate 2004-01-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9BC43
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ167V0
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8P126
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5Y8S5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8ZV53
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5M0B8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7J0M3
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2SEZ5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5Y8Y0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5UF74
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP54363
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9AF06
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ47XQ8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3N5L9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7V7D8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5YDB0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5M216
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD5VT38
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1JM38
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID15613034
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID11886
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2FG92
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2SHR3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8Z8T4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22498
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD7DQT8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5M3Y6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ17W08
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9AYX1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8NVG5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7IEY2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06850
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6MHW4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VAL5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5I6E1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8ZC94
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD7E9E7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7IIS0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3251
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5M4W5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP44309
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2G5F0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DB96
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373802
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9GFF3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9HPQ9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID44999375
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DB97
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1JC56
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP44317
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6LT81
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0MAM5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VRB8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09057
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ12W31
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9HEW1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2JCQ7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5Y0N8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5LUY8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409261251
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7JPZ4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1WDB0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6LTE9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2GAK1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3MYY8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD3ZQL7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9I0U7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ47N45
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423545303
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP77989
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395152
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16132357
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5GSL0
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID37602
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5LZD4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID519017
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9BG28
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2YAI3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1JH84
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6LZG8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7JVC2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22251485
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0CZ62
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5FKY7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ91082
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2FXU0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6M0X3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3PE89
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0CZ63
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100136771
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5HY32
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ83M42
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD5E7U7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19402
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2IU50
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VKQ4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP78599
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1GTG6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP43856
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VLH2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ44233
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5NH50
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID378608
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1GYN9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22923
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID406259
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2118
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ90029
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ12LL4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO60109
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP75119
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395120
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5NII9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ90033
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2W3C2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1U4H0
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423545302
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VQZ6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID9924867
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8YVP7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22649
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6HAV3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5ITF9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC6E585
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7JHF2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP75388
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3NRB5
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID10245
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5M6K8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1GE59
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC6BSW0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1148
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5IZD7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ145V4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2YT95
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06219
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6GJG1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DD40
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5N1I0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06296
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DD41
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC6DB82

Total number of triples: 1428.