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filingDate 2004-02-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fe771e5d54b82a018652fe9857a38d8e
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7bb233e9b092ee00d36e5e77fa9e51c2
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publicationDate 2005-11-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1597585-A2
titleOfInvention Method for selecting a candidate drug compound
abstract The invention relates to the field of candidate drug testing and drug development. A method is provided for providing a compound composed of at least one molecule attached via at least two linkages to a molecular scaffold, said method comprising providing a scaffold comprising at least a first and a second reactive group; providing at least one molecule capable of reacting with said at least first and second reactive group; contacting said scaffold with said at least one molecule to form at least two linkages between said scaffold and said at least one molecule in a coupling reaction, whereby the formation of a linkage accelerates the formation of a consecutive linkage, preferably wherein said coupling reaction is performed in solution, more preferably in an aqueous solution. Furthermore, a method is provided for selecting a candidate drug compound, comprising providing a library of compounds according to the invention and determining the binding of a target molecule to said compounds.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2651964-A2
priorityDate 2003-02-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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