http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1442022-A2

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filingDate 2002-11-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_12514504a6dafd1312954741267e7496
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publicationDate 2004-08-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1442022-A2
titleOfInvention Polyamide modulators of cox2 transcription
abstract Processes and compositions are provided for regulating COX2 gene expression in a cell. The process includes selecting a polyamide composition comprising N-methyl pyrrole (Py) and N-methyl imidazole (Im) to provide specific binding to DNA at a COX2 gene target site in a cell. The polyamide is then combined with the cell containing the COX2 gene, wherein the polyamide binds to the COX2 gene promoter target site and regulates transcription of the COX2 gene.
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