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filingDate 1997-09-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6fd5b3c94116c0922ec21b0aef685a61
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publicationDate 2004-06-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1424069-A2
titleOfInvention Gastric-retentive, oral drug dosage forms for the controlled-release of sparingly soluble drugs and insoluble matter
abstract Controlled-release oral drug dosage forms that comprise a tablet or capsulencontaining a plurality of particles of a solid-state drug dispersed in answellable/erodible polymer, such as poly(ethylene oxide) are described. Onceningested, the tablet or capsule disintegrates to disperse the particles within thenstomach where they imbibe water to cause them to swell and promote retention innfed-mode-induced patients. As the gastric-retained dosage form gradually erodes, thendrug is released in a controlled manner to the stomach for treatment of localndisorders, and to the upper gastrointestinal tract where it becomes available fornabsorption in a controlled and therapeutic manner. Drug containing vesicles, such asnliposomes or nanoparticles or enteric-coated drugs particles, can also be delivered tonthe gastrointestinal tract in a controlled manner using the gastric-retentive dosagenforms of the present invention.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14969
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP70160
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419533490
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81423
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419533562
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5546
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492026
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81497
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09476
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67973
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4173
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54675776
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67971
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5PJB2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226411901
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67974
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129515347
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID52330067
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24241
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67968
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419491958
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408598248
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67970
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67969
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129741655
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419581777
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCH0ZG98
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5IGQ0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01262
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5755
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11245343
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81025
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01261
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396738
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128856633
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13135
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID796
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226416540
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4T554
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01258
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ98TA8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226416539
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01257
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13190
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01260
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01259
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419560480
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9TQY7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2XNF5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419533778
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3639
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12040205
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226416538

Total number of triples: 358.