http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1418945-A2

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_d05c497d8397361b0b709dbede445d68
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-6907
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-22
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-48
filingDate 2002-03-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_31de12d72d1eab75ac0f775f359d991b
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4306e240e7ef5609d4dc2b8f9c8501df
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_265999fde422e8784c68dc9dabe1d081
publicationDate 2004-05-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1418945-A2
titleOfInvention Micellar drug delivery vehicles and uses thereof
abstract Anhydrous formulations are formed of a diblock copolymer (X-Y) having a hydrophilic bloc X comprising residues of monomer x, and a hydrophobic block Y comprising residues of monomer y; an additive selected from a polymer and an organic solvent, where the solvent is water-miscible and biocompatible, and the polymer is hydrophobic or hydrophilic and comprises residues of monomers x and/or y, the polymer optionally having a molecular weight that is less than the molecular weight of the diblock copolymer; and a drug. Upon admixture with water, the anhydrous formulations form drug delivery vehicles, preferably in micellar form. The inclusion of polymer and/or organic solvent provides for the formation of micelles at an enhanced rate, and/or provides the formation of micelles having an enhanced ability to incorporate drug(s), and/or provides the formation of micelles having advantageous physical characteristics, e.g., advantageous viscosity and/or melting point.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-6699694-B1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-7732164-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2013156944-A1
priorityDate 2001-03-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 447.