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http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_05a203d85ee01909eaf728dc16f0f6cb
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D213-57
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D217-06
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D213-57
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B61-00
filingDate 2002-07-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2006-04-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3df12f11034175fd9503f38f796c13b8
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d495ed53ba9ed9aa70a6263e7099b7fa
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d41b2ee185e6ed01204e5cb66140d028
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a3e7a0f953be13ddb42a28bee7a5c80e
publicationDate 2006-04-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1412331-B1
titleOfInvention Process for the production of 4-amino-2,5-bisheterocyclylquinazolines
abstract The invention provides a process for the production of a compound of formula (A), or a pharmaceutically acceptable salt or solvate thereof, wherein R1 represents C¿1-4? alkoxy optionally substituted by one or more fluorine atoms; R?2¿ represents H or C¿1-6? alkoxy optionally substituted by one or more fluorine atoms; R?3¿ represents a 5- or 6-membered heterocyclic ring which is optionally substituted; R4 is a 4-, 5-, 6- or 7-membered heterocyclic ring which is optionally fused to a benzene ring or a 5- or 6-membered heterocyclic ring, the ring system as a whole being optionally substituted; the process comprising condensing a compound of formula (B), wherein R1 to R3 are as defined above; with a compound of formula (C), wherein R?5 and R6¿ taken together with the N atom to which they are attached represent a 4-, 5-, 6-, or 7-membered N-containing heterocyclic ring, the ring being optionally fused to a benzene ring or a 5- or 6-membered heterocyclic ring, the ring system as a whole being optionally substituted.
priorityDate 2001-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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