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filingDate 2002-06-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7f4c0744b7c30bb70d2e929c9ecd7d71
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publicationDate 2004-04-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1405644-A1
titleOfInvention Tissue-specific transporter inhibitor
abstract The present invention is to provide a tissue-specificntransporter inhibitor which is not absorbed through thendigestive tract and can prevent deterioration in the QOL of anpatient caused by diet therapy, and a therapeutic drug forntissue dysfunction diseases and a therapeutic drug fornsuppressing the progress of chronic renal failure containingnthe inhibitor as an active ingredient. A tissue-specificntransporter inhibitor which is not absorbed through thendigestive tract is constructed by introducing a dipeptide whichnis a ligand of an oligopeptide transporter 1 into ansupramolecular structure polyrotaxane wherein itsnstructurally modified active residue is expected to benexcellent in the interaction with a transmembrane transporter.
priorityDate 2001-06-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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