| abstract |
The present invention provides an anilinenderivative represented by the formula (I)n nwherein R 1 and R 2 are each H, (C 1-12 )alkyl, (C 3-8 )cycloalkyl,nhydroxy (C 1-12 )alkyl , hydroxycarbonyl (C 1-12 )alkyl, (C 1-6 )-alkoxycarbonyl(C 1-6 )alkyl,n-COR 8 , wherein R 8 is H, halo-(C 1-12 )alkyl,n(C 3-8 )cycloalkyl or (substituted) phenyl, COOR 9 ,nwherein R 9 is a halo(C 1-6 )alkyl group, (substituted) phenylnor (substituted) benzyl; R 3 , R 4 , R 5 , R 6 and R 7 are eachH, halogen,nOH, nitro, halo(C 1-12 )alkylthio, (substituted) amino-(C 1-2 )alkyl,n(substituted) phenyl, (substituted) benzyl,namino, -N(R 10 )R 11 wherein R 10 and R 11 are each H, alkyl,ncycloalkyl, (substituted) phenyl, (substituted) benzyl,n-COR 8 or COOR 9 , or (C 2-27 )perfluoroalkyl, etc., and a processnfor producing the aniline derivative. According to thenprocess of the present invention, perfluoroalkylanilinenderivatives can be obtained by using various anilines as thensubstrate with a high position selectivity and high yield. |