http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1377582-A1

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filingDate 2002-04-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_966589e96dfc506e5379fe3919eb242f
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5d95a5a75b9d0acbd454fbe8f51d485e
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d5619df7c3b1948c54ebd0f058289160
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_836c1377ba17debe7093ca29835335bb
publicationDate 2004-01-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1377582-A1
titleOfInvention Novel 3-c(o)r substituted 10-cyclohexylbenzoyl pyrrolobenzodiazepines; tocolytic oxytocin receptor antagonists
abstract The present invention provides novel tricyclic benzodiazepine carboxamides compounds and methods and pharmaceutical compositions utilizing them for the treatment and/or prevention and/or suppression of disorders which may be remedied or alleviated by oxytocin antagonist activity, including prevention and/or suppression of preterm labor, suppression of labor at term prior to caesarean delivery, and for the treatment of dysmenorrhea. These compounds are also useful in enhancing fertility rates, enhancing survival rates and synchronizing estrus in farm animals; and may be useful in the prevention and treatmraent of disfunctions of the oxytocin system in the central nervous system including obsessive compulsive disorder (OCD) and neuropsychiatric disorders.
priorityDate 2001-04-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 695.