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filingDate 2002-01-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2003-12-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1365754-A2
titleOfInvention Inhibition of proteasomes to prevent restenosis
abstract Restenosis of blood vessels after angioplasty is achieved by preventing of cell proliferation, particularly of smooth muscle cells, in blood vessel walls by inhibiting the ubiquitin-proteasome protein degradation pathway. The inhibition is accomplished by administering to the cells in the blood vessel walls a compound, e.g., a protein or small molecule, capable of inhibiting the ubiquitin-proteasome protein degradation pathway. The inhibiting compound is preferably administered by coating the compound on a stent and implanting the stent in the blood vessel after angioplasty.
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