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filingDate 2001-09-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1acafa3673eb5af7be3e23e75e6ce87d
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publicationDate 2003-07-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1330470-A1
titleOfInvention Glutathione conjugates with distamycin derivatives having antitumor activity
abstract The present invention refers to distamycin and derivatives thereof, such as bromo-or chloro-acryloyl derivatives of distamycin, which are conjugated with glutathione, to a process for their preparation and to pharmaceutical compositions thereof. The compounds of the invention are endowed with a remarkable antitumor activity and are thus useful in therapy in the treatment of cancer.
priorityDate 2000-09-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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