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filingDate 2002-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0714dd3683d14d9f7a5128b41b3fc286
publicationDate 2003-02-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1284257-A2
titleOfInvention Difluoromethylene aromatic ethers and their use as inhibitors of the glycine type-1 transporter
abstract This invention relates to a series of difluoromethylene aromatic ethers of the formulan nwherein ring A and X and Y are defined as in the specification, that exhibit activity as glycinentransport inhibitors, their pharmaceutically acceptable salts, pharmaceutical compositionsncontaining them, and their use for the enhancement of cognition and the treatment of thenpositive and negative symptoms of schizophrenia and other central nervous system disordersnin mammals, including humans.
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Total number of triples: 428.