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filingDate 2000-11-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e8102dc0673ea27b431f8bd46425956b
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_71974bec34ff338deea040ca6f487b04
publicationDate 2002-09-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1235922-A2
titleOfInvention Excipient system that contains coating substances with enzymatically removable side-groups
abstract The invention relates to an excipient system that can be obtained by (1) optionally mixing a component a2) with a component a1) in a molar ratio [a2):a1)] of 1:1 to 1000:1, preferably between 10:1 and 100:1, (2) mixing the complex resulting from step (1) or the complex a1) alone with a component b1), preferably in a molar ratio b1):a1) + optionally a2) of 1:1 to 1:1000, said mixing ratio being adjusted in such a manner that the net charge of the resulting total complex is preferably neutral or anionic. Component a1) comprises an active substance a1), a binding structure a1) for the binding structures b1) or a2), wherein the active substance a1) may contain the binding structure a1). Component a2) comprises a binding structure a2) for the binding structure a1) and a carrier a2) which may contain the binding structure a2). Component b1) may comprise a binding structure b1) for the binding structure a1), for the active substance a1), for the binding structure a2) or for the carrier a2), a coating substance that may contain the binding structure b1), an enzymatically removable connector, and an anionic side-group. The invention further relates to the production and to the use of the inventive excipient system.
priorityDate 1999-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 570.