http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1181009-A1

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filingDate 2000-05-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d10290fdecc17fde556930dbaf1e39e7
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1da85047759a85afdd851f162f14e3b9
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_568ca9e738910d912d7f01acb27f07a9
publicationDate 2002-02-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1181009-A1
titleOfInvention Method of producing submicron particles of a labile agent
abstract The present invention relates to a sustained release composition comprising micron particles of labile agent and a method of preparing and using the sustained release composition. The invention further relates to micron particles of a labile agent and a method of preparing the micron particles. The method of the invention for preparing a composition for the sustained release of a labile agent, comprises forming a suspension comprising the labile agent dispersed in a polymer solution comprising at least one biocompatible polymer and at least one polymer solvent. The suspension is then wet milled to achieve micron particles of the labile agent. The polymer solvent is then removed resulting in a solid polymer/labile agent matrix. The composition for sustained release of a labile agent is likewise prepared according to the method of the invention. The sustained release composition of the present invention can be used in a method for providing a therapeutically effective blood level of a labile agent, in a subject in need of treatment with said agent, for a sustained period comprising administering to the subject the sustained release composition described herein. The method for preparing micron particles of a labile agent comprises forming a suspension comprising the labile agent, dispersed in a polymer solution comprising at least one biocompatible polymer and at least one polymer solvent, and wet milling of the suspension. The submicron particles of labile agent, as described herein, are prepared according to this method.
priorityDate 1999-05-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP34747
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP18109
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6YK33
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP34746
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJI1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419562219
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8617806
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10112
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP58343
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419524130
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJI4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1245926
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21989438
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJU0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13190
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13529
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJT9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO70615
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1255582
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID986791
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410511156
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11535
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ91082
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13391
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCE3YBA4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3FFS8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73848
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06297
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID18976
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP58756
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73727
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23830
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ05163
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID679
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73849
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5IGQ0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8HYE5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5360315
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87059419
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24335
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8615933
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID36878
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3169327
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48248
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID57569658
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3474008
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559095
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11885
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11029
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129049279
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID44544175
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID39251
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67930
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1HFN3
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226410154
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6212
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419537701
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20391
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO62754
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67931
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GKA1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID105090400
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1403863
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID378781
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67968
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403795

Total number of triples: 377.