http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1173602-A1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_2a819eda0adf22936a52362eeebb9fb4
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K14-811
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K14-81
filingDate 2000-04-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9488202991bd45aab648ad3d2c1df427
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6d6a6d5a8f12d21b7956536063e6bfa5
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bc2a1d19d9caa6d935ed55c2ad949d59
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_317b20b0c2b29231724677d97c3d50c5
publicationDate 2002-01-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1173602-A1
titleOfInvention Ecotin derivatives
abstract This invention provides a class binding proteins that specifically bind to and modulate (e.g. enhance) the activity of polypeptides having a chymotrypsin fold (e.g. serine proteases). The binding proteins are based on the structure of ecotin. It was discovered that modification of the amino or carboxyl terminus and/or randomization of one or more of loops 50s, 60s, 80s or 100s will provide an ecotin variant library from which can be selected binding molecules (e.g. protease modulators) specific to virtually any serine protease. Depending on the ecotin variant and the target serine protease, the modulator can act as a serine protease inhibitor or as a serine protease activator. Specific agonists (enhancers) of Factor IXa are disclosed.
priorityDate 1999-04-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2UVH8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID493738
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WN82
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2TBU0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5RF29
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WN83
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419490256
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9I9M4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID26101581
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6274
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281408
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9IB11
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP17721
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9I9L5
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11287
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394420
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ97BJ8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07628
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID738078
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP57384
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81800
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419483812
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCG1K2D9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419490523
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ37875
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69159
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID108180329
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373313
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69160
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP34129
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09537
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2056
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2KJ63
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID85253
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07647

Total number of triples: 678.