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filingDate 2000-03-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_293d1e9d879599914dcc37195f6e67aa
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fbe3aa3fb65f8a7b92ac878c72b7edb3
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6d444af9620aa70f72e4d575975b59c4
publicationDate 2002-01-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1165528-A1
titleOfInvention Novel morpholine derivatives, method for the production thereof and pharmaceutical preparations containing said derivatives
abstract The invention relates to compounds of formula (I) and the salts thereof with mineral or organic acids, the solvates and/or hydrates thereof, exhibiting a strong affinity and high degree of selectivity with respect to human NK1 receptors of substance P. The invention also relates to a method for the production of said derivatives, intermediate compounds of formulae (IV), (VI) and (VIII) used in the production thereof, pharmaceutical compositions containing said derivatives and the use thereof in the production of medicaments in the treatment of all pathologies where substance P and/or human NK1 receptors are involved.
priorityDate 1999-03-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6865
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID232361682
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6863
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID232364669
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128144183
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID404136
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID81531
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID232364644
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO13465
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID17934368
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID232363900

Total number of triples: 312.