| abstract |
The present invention relates to new highly functionalized heterobicyclenderivatives of following general formula (I), prepared by a process which involvesnonly two steps by using, as starting products, commercially available, or easilynprepared, α-amino ketones and α,β-dihydroxy acids or α-amino-β-hydroxy acidsnor α-hydroxy-β-amino acids or α,β-dithiol acids derivatives and to librariesncontaining compounds of formula I and to the generation of such combinatorialnlibraries composed of compounds of formula I, in individual synthesis, mixturensynthesis, split and recombine synthesis and parallel synthesis either in manual ornautomated fashion. |