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filingDate 1999-06-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1ad59413576bd715db9978bde88ee3ce
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_42293061464539adf20a4cacd6143a46
publicationDate 2001-05-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1094800-A2
titleOfInvention PEPTIDYL-PROLYL $i(CIS)-TRANS ISOMERASE INHIBITORS AND USES THEREFOR
abstract The invention relates to inhibitors of PPIase activity and pharmaceutical compositions containing such inhibitors. Such compounds are useful for treatment of disorders characterized by inappropriate cell proliferation. In particular the compounds disclosed herein inhibit the activity of members of the Pin1/parvulin class of PPIases. These compounds have been designed based on the high resolution X-ray derived crystal structure of the human enzyme Pin1.
priorityDate 1998-06-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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