http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1054868-B1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_afc5d8c9ee6673323cee3e2d19bc5146
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D213-82
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-00
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P13-08
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D213-82
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P43-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-497
filingDate 1999-02-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2003-09-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c2929e3fa1e4e06918c24599f767fc49
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0503072c90838a73d4befe2fc3c3bd88
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_58212e8ff1b6f3a50ea1d3e101763c3d
publicationDate 2003-09-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1054868-B1
titleOfInvention Substituted pyridino arylpiperazines useful in the treatment of benign prostatic hyperplasia
abstract This invention relates to a series of heterocyclic substituted piperazines of Formula (I), methods of treatment, pharmaceutical compositions containing them, and intermediates used in their manufacture. The compounds of the invention selectively inhibit binding to the α-1a adrenergic receptor, a receptor which has been implicated in benign prostatic hyperplasia. As such the compounds are potentially useful in the treatment of this disease.
priorityDate 1998-02-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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