http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0910416-A2

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filingDate 1997-06-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_cc82991623131748f0937b9cf8bc5e36
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e3e0228a61e4c2326890a2b57cec6dfa
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5e658872c880cc34b4a6e7cb2c972b4f
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f9fe724a5a71133dcea76512fa546003
publicationDate 1999-04-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0910416-A2
titleOfInvention Radiopharmaceutical compositions capable of localizing at sites of thrombus
abstract A radiopharmaceutical capable of localizing at a site of thrombus containing activated platelets within a mammalian body is provided wherein the radiopharmaceutical comprises a linear peptidomimetic containing ligand capable of specifically binding to the GPIIb/IIIa integrin receptor of platelets in the thrombus and a radionuclide covalently bound to the peptidomimetic containing ligand. The ligand compositions of the invention are provided complexed with a selected metal radionuclide to form a diagnostic or therapeutic radiopharmaceutical to image a site of thrombus or provide radiotherapy to the site of thrombus, respectively. Methods of imaging a site of thrombus in a mammalian body by administering a diagnostically effective amount of the radiopharmaceutical composition of this invention complexed with a selected diagnostic metal radionuclide and methods of providing therapy to a site of thrombus in a mammalian body by administering a therapeutically effective amount of the radiopharmaceutical composition of this invention complexed with a selected therapeutic metal radionuclide are also provided as well as kits for preparing such radiopharmaceutical compositions.
priorityDate 1996-06-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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