http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0822812-A4

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filingDate 1996-03-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_824c0344b50cdf76a76f75c5486b784b
publicationDate 2000-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0822812-A4
titleOfInvention LOCAL TREATMENT AND / OR PREVENTION OF SUBCUTANEOUS SOCUS AND OVERLAYING SKIN TISSUE USING ACETYLCHOLINE PRE-STAGES AND CATECHOLAMINES
abstract Compositions for the topical treatment of sagging subcutaneous muscle and overlying cutaneous tissue contain catecholamines and/or related compounds in a dermatologically acceptable carrier. Examplary catecholamines include adrenaline, norepinepherine, dopamine and their precursors; catecholamine precursors such as tyrosine and phenylalanine are preferred. Preferred embodiments further contain at least one other ingredient that enhances neurotransmitter synthesis and/or skin penetration. In some embodiments, an acetylcholine precursor such as dimethylaminoethanol and/or a fatty acid ester of ascorbic acid are included in the formulation. In these and other embodiments, particularly those employing tyrosine and/or phenylalanine as a catecholamine precursor, other cofactors such as vitamin B6 and pantothenic acid or calcium pantothenate are included in the composition to enhance the action of the active ingredients. Other compounds that scavenge free radicals and antioxidants may also be added.
priorityDate 1995-04-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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