Predicate |
Object |
assignee |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_fd569fbfa1953ca9b7b375510e4d2763 |
classificationCPCAdditional |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C2601-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C2601-08 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D295-13 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D213-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C231-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C233-36 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D265-30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07B53-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C215-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D295-125 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-44 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C231-18 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C231-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C215-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C233-36 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D211-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D295-13 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D295-125 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D211-44 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B53-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C231-18 |
filingDate |
1996-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate |
2003-09-03-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1206061fb9aebaceced1bd640759bde8 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4701b544fc14308af430389c445dc2cb http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_86042162fb4f8fd8c1a29d388042cecd |
publicationDate |
2003-09-03-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
EP-0782992-B1 |
titleOfInvention |
Amino alcohol derivative and method for preparing the same |
abstract |
A process for preparing a 2-acylamino alcohol derivative which comprises (A) reacting an aminopropanol derivative represented by the following formula (1): Y-CH2-C*H(NHP<1>)-C*H(OH)-R<1> with an amine represented by R<2>H to synthesize an amino alcohol derivative represented by the following formula (2): R<2>-CH2-C*H(NHP<1>)-C*H(OH)-R<1> (B) leaving P<1> from said amino alcohol derivative represented by formula (2) to synthesize an amino alcohol derivative represented by the following formula (3): R<2>-CH2-C*H(NH2)-C*H(OH)-R<1> (C) reacting said amino alcohol derivative represented by formula (3) with a carboxylic acid represented by R<11>COOH or a reactive derivative thereof to prepare a 2-acylamino alcohol derivative represented by the following formula (4): R<2>-CH2-C*H(NHCOR<11>)-C*H(OH)-R<1> wherein * represents an asymmetric carbon atom, and P<1>, R<1>, R<2> and R<11> are defined in the specification. A process for preparing alcohol derivatives having an acylamino group through several steps from amino group-protected 2-aminopropanol derivatives, and novel amino alcohols useful as intermediates in the process for preparing the alcohol derivative. |
isCitedBy |
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10927092-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10227323-B2 |
priorityDate |
1995-12-08-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |