http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0730582-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_1c89ce4d9ac03f9acd8ddede1162f94d |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D261-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D231-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D261-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 |
| filingDate | 1994-11-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9ea117a3d1498dd06fdb65e4fb38136c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_21530588924af8d92d24b2e681584290 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0e0c2fc3012d4c5ffbe36101aa03b611 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_643d53713ada9541106f418ed0e8c9e8 |
| publicationDate | 1996-09-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | EP-0730582-A1 |
| titleOfInvention | Isoxazole and pyrazole derivatives as dopamine receptor subtype ligands |
| abstract | A class of substituted isoxazole and pyrazole derivatives of formula (I), or a salt thereof or a prodrug thereof, wherein the broken circle represents two non-adjacent double bonds whereby the five-membered ring containing X and Y is aromatic; one of X and Y represents nitrogen, and the other of X and Y represents oxygen or N-R5; R1 represents hydrogen, C¿1-6? alkyl or trifluoromethyl; R?2 and R3¿ independently represent hydrogen, hydrocarbon, a heterocyclic group, halogen, cyano, trifluoromethyl, nitro, -OR?a, -SRa, -SORa, -SO¿2Ra, -SO2NR?aRb, -NRaRb, -NRaCORb, -NRaCO¿2R?b, -CORa, -CO¿2Ra or -CONRaRb; R4 represents hydrocarbon or a heterocyclic group; R5 represents hydrogen or C¿1-6? alkyl; and R?a and Rb¿ independently represent hydrogen, hydrocarbon or a heterocyclic group, are ligands for dopamine receptor subtypes within the body and are therefore useful in the treatment and/or prevention of disorders of the dopamine system, in particular schizophrenia. |
| priorityDate | 1993-11-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 387.