http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0726761-B1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_880ee63bc25f3bfd79814fac88158ca2
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-1075
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-113
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-113
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-107
filingDate 1994-11-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2001-01-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bbcac52a25e64b2442df58f3f29d7c2e
publicationDate 2001-01-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0726761-B1
titleOfInvention Microparticular pharmaceutical compositions in micellar form
abstract A pharmaceutical composition comprises microparticles in micell. The microparticles contain at least one pharmaceutically-active agent, at least one water soluble or miscible phospholipid, at least one lipid soluble or miscible phospholipid, at least one non-ionic surfactant having an HLB value of about 15 or greater, at least one non-ionic surfactant having an HLB value of about or less, and at least one water soluble or miscible sterol compound. The microparticles are suspended in at least one fatty acid having a chain length of C14 or less. The composition may optionally contain at least one fatty acid having a chain length of C16 or greater in a concentration of about 5 w/v % or less. The composition is prepared by admixing the pharmaceutically-active agent, phospholipids, surfactants, and sterol, micronizing the admixture to form microparticles, and suspending the microparticles in at least one fatty acid of chain length of C14 or less to form microparticles in micell. The invention may be useful in the oral administration of drugs and other therapeutic agents, as well as for the trans-umbilico-dermal administration of such drugs and therapeutic agents.
priorityDate 1993-11-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0CP75
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP37886
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JAX9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48248
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JAY0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JAY1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395375
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB32
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129289952
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128780205
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9852308
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GMB2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB33
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128387026
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GMB3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB34
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB35
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11005
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6750
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396570
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18667284
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB36
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID644119
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09476
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB37
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID841689
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09477
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB38
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14985
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403426
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB39
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID151056
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ56JA9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB24
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396279
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09537
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397879
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GKA2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB25
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31307
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID665270
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB26
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395359
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20391
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GL60
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB27
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20392
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67968
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB28
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID136079170
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14455022
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129573886
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67969
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB29
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67970
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81423
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB30
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67971
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB31
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10224496
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID378781
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67973
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB16
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9924977
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21585014
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ68VT0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67974
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397717
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB17
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP55755
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399496
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5BMR2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB18
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16218600

Total number of triples: 1024.