http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0725795-A1

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filingDate 1995-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_36e96a1a0656fd4ba6a922f32729c868
publicationDate 1996-08-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0725795-A1
titleOfInvention Single-chain forms of the glycoprotein hormone quartet
abstract Single-chain forms of the glycoprotein hormone quartet, at least some members of which are found in most vertebrates, are disclosed. In one embodiment of these single-chain forms, the alpha and beta subunits of the wild-type heterodimers or their variants are covalently linked, optionally through a linker moiety. A drug may further be included within the linker moiety to be targeted to receptors for these hormones. Some of the single-chain forms are agonists and others antagonists of the glycoprotein hormone activity. Another embodiment of the single-chain compounds of the invention comprises two beta subunits of the glycoprotein hormones, which beta subunits are the same or different. These "two- beta " forms are antagonists of glycoprotein hormone activity.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014159813-A1
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type http://data.epo.org/linked-data/def/patent/Publication

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