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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D497-20
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filingDate 1995-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7b38d5c67a81e2a3ddf82e0dbf0565bb
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a8da24ccdcd8ec54ee0d27d56735ec30
publicationDate 1996-01-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0689836-A1
titleOfInvention Spirooxathiolane-quinuclidine derivative for the treatment of xerostomia
abstract A therapeutic agent for the treatment of xerostomia comprises a derivative of spirooxathiolane-quinuclidine or an acid addition salt thereof as an active ingredient represented by the following formula [I]:n n (wherein R¹ and R may be the same or different and each represents hydrogen, alkyl, cyclopentyl, cyclohexyl, aryl, diarylmethylol, or alkyl which may be substituted by one or more aryl groups). n The above therapeutic agent can be administered orally or parentally and cure xerostomia. Specifically, the agent can be used for improving and/or curing dry mouth caused by various diseases with organic changes in salivary gland, lesions in salivary gland accompanied with systemic diseases, necrosis of salivary gland cell by radiotherapy, HIV infection (AIDS), hypo-function of saliva secretion, affection of various medicines taken and, further, mental fatigue or bad conditions due to complex social life situations.
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priorityDate 1994-06-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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