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filingDate 1992-05-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 1995-11-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0586523-A4
titleOfInvention Determination of prodrugs metabolizable by the liver and therapeutic use thereof
abstract A method of ascertaining if a prodrug is useful for treating a disease is disclosed. The prodrug is acceptable if it is metabolized in liver cells by aldehyde oxidase to produce an active drug or metabolite. Prodrugs are shown equally effective in treating diseases as the active drug itself with many benefits and without as many associated side effects. Methods for treating cancers with 5-iodo-2-pyrimidinone-deoxyribose and 5-fluoro-2-pyrimidinone are also described.
priorityDate 1991-05-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2VH51
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9MTJ2
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7MNI9
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00326
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9VPT7
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0KCB9
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCE1ACQ9
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4T4H1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0R541
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1U4L8
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237945958
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226937135
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7MVK1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9P6C8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70269
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DOM8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP05336
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8G1S6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID102197
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9P4C2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DOM7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP85440
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8AJ16
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237966369
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1890
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9AW39
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19971
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8HA92
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0HQ66
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4TH00
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9MCL2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ884R6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID38871
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9444
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9KV80
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ12D54
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID20322
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID928935
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2I2C4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ483R6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID65161
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67812859
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2FKG1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135594056
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2SD94
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415804679
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4SMV5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2K6P6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ12P69
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ21KC3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4SP57
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VLH2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4REE0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0HLE9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226937134
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4TC44
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6275
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66308
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8LEB2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426086920
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4SZJ3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68466386
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID238090297
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8XWC2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4SRU3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0V9X6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3707550
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VQZ6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21117604
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID238260666
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0TM56
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121698
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5E7J6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419585666
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1870
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1J2Q5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ12QG2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413552893
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0HNM4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ99N42
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP86883
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0VPV2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1KP56
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1201441
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP86885
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1JH60
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3M1J3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3K0G3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0DWH1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP86884
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2A3D8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226425245
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID79655
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1H0L2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ31ZS8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226434941
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1VUR5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67816414
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7HKJ0
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226434940
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57228359
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ21UZ9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7NI79
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7HCC9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453861888
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2656999
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0HXQ3
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456171974
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4TU42
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70799353
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7IF30
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06478
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP93629
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7I271
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450423200
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7JI79
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ609M6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06525
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID23778904
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1201482
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7ISJ1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1UY21
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7VMU2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7V3J3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP89446
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7CP66
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5F068
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4TQT5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6478043
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID381087
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5QX61
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419587275
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8EHK3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5FP57
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5P0Z5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ32GW8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3MAQ6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5XZ80
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0ITW7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419505951
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5R757
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ88F51
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7GUU5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Q8N6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB6ERX7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC1DJM5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8NXU1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0RM77
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB3E2L0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7Z9S5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3K803
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67152712
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC1EN92
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3LLP9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4593165
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8P126
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3L983
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC5C4W6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5148055
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ55DV9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID649
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415806783
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3P4M1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70265
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8E3L7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4TZG4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8CGY4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14281
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID60923442
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453940049
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ48KQ0
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID239393571
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8II06
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8NVG5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8H2R9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21518
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9JDB9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9IUG9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70807678
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2I2L6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID117607474
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1269845
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54267272
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0PWX8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ54TC2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ38WJ3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9K286
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126941

Total number of triples: 1823.