http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0522868-A1

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filingDate 1992-07-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_aa78a42ba3d19869c8ebadc9ebf9b732
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publicationDate 1993-01-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0522868-A1
titleOfInvention A human endothelin receptor
abstract DNA encoding an endothelin receptor shown in SEQ ID NO: 1 or 2 in the Sequence Listing is isolated from cDNA which is prepared from poly(A)⁺RNA derived from a human placenta. In addition, an expression vector containing the DNA and a transformant containing the expression vector are obtained. An endothelin receptor is obtained by culturing this transformant. A receptor shown in SEQ ID NO: 1 is an ET A -receptor which has a high affinity for endothelins 1 and 2, especially for the endothelin 1. A receptor shown in SEQ ID NO: 2 is an ET B -receptor which has an affinity for endothelins 1, 2 and 3 with no selectivity.
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