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filingDate 1990-08-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 1991-03-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0418597-A2
titleOfInvention Controlled release carbonic anhydrase inhibitor containing pharmaceutical compositions from spherical granules in capsule oral dosage unit form
abstract A controlled release pharmaceutical composition in oral dose unit form comprising a hard or soft shell capsule containing a filling comprising a therapeutically effective number of active spherical granules comprising an effective amount of at least one carbonic anhydrase inhibitor active medicament, a pharmaceutically acceptable normally solid diluent adapted to form a diffusable matrix for the carbonic anhydrase inhibitor active medicament and an optional pharmaceutically acceptable excipient. A method for the preparation and for the administration of the above defined composition is provided as well.
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