| abstract |
Inhibitors of phospholipase A 2 activity at the cell-surface membrane whose molecular structure comprises a cell-permeable PLA z -inhibitor moiety covalently bonded directly or indirectly to a physiologically acceptable carrier moiety which is effective to inhibit cell internalisation of the cell-permeable PLA 2 -inhibitor moiety, with the proviso that phosphatidylserine is not bonded indirectly via divalent dodecanedioyl to dextrane hydrazide. |