http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0213481-A3
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K38-00 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K5-06078 |
| classificationIPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K38-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K5-065 |
| filingDate | 1986-08-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 1989-07-19-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | EP-0213481-A3 |
| titleOfInvention | N-terminally substituted dipeptide amides no. 2 |
| abstract | This invention encompasses compounds of the formula n nand the pharmaceutically acceptable acid addition salts thereof nwherein R¹ is lower alkoxy or -O-(CH₂) n -phenyl where the nphenyl may be optionally substituted with halogen, -NO₂, -CN, n-NH₂ or lower alkyl wherein n is 1 to 4; R² and R³ nrepresent lower alkyl, halogen, lower alkoxy or one of R² or nR³ is hydrogen and the other is lower alkyl, lower alkoxy, or nhalogen; R⁴, R⁵, R⁷, R⁸, and R⁹ represent hydrogen or nlower alkyl, R⁶ represents hydrogen, lower alkyl, lower nalkenyl, or -(CH₂) m -cycloalkyl wherein m is 1 to 4 and the ncycloalkyl has 3 to 8 carbon atoms; R¹⁰ is -(CH₂) p -phenyl nwherein p is 1 to 4; and v represents an asymmetric carbon that nmay be racemic or have the D or L Configuration; nw represents an asymmetric carbon when R⁷ and R⁸ are not nthe same that may be racemic or have the D or L configuration. nThis invention also encompasses compounds where R¹ is nhydroxy, provided at least one of R⁴, R⁵, R⁶ or R⁹ is nlower alkyl. The compounds of this invention are useful nanalgesic agents. |
| priorityDate | 1985-08-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 22.