http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0131006-A1
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_46443201668cc985a4ce2fb287770f99 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D285-10 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-535 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-41 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D- http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D285-10 |
filingDate | 1983-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f1e2a4d7da2f408b3b173f242d0dd433 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_21e986be17c326d4469bcf839d1d5aa6 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a0f7ffb75855c2b14806843216a9e540 |
publicationDate | 1985-01-16-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | EP-0131006-A1 |
titleOfInvention | ESTERS OF DERIVATIVES OF 1,2,5-THIADIAZOL 3- (3-SUBSTITUTE-AMINO-2-HYDROXYPROPOXY) -4-SUBSTITUE. |
abstract | New compounds of formula (I) where R is lower alkyl, lower cycloalkyl, lower haloalkyl, lower alkylcarboxymethyl, arylcarboxymethyl, lower alkenyl, lower alkynyl, aryl having between 6 and 10 carbon atoms, or an aralkyl; R1 is lower alkyl, lower hydroxyalkyl, lower alkenyl, lower alkynyl, aralkyl or -WB; where W is an alkylene containing between 1 and 10 carbon atoms and B is -NR2COR3, -NR2CONR3R4, -NR2SO2R3, -NR2SO2NR3R4 or -NR2COOR5, where R2, R3, R4 and R5 may be the same or different and may be hydrogen, a alkyl, alkoxyalkyl, alkoxyaryl, cycloalkyl, alkenyl, alkynyl, aryl, etheroaryl, or aralkyl, provided that R3 and R5 are not hydrogen when B is -NR2SO2R3 or -NR2COOR5, or R3 and R4 can form with N a heterocyclic group comprising from 5 to 7 elements; A is a direct bond, a lower alkylene or a lower alkene having between 1 and 10 carbon atoms; as well as their pharmaceutically acceptable salts. These compounds are useful as beta-adrenergic blocking agents and for the treatment of glaucoma. |
priorityDate | 1982-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 291.