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http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D281-10
filingDate 1982-07-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 1984-01-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0098892-A1
titleOfInvention Process for preparing 1,5-benzothiazepine derivatives
abstract A process for preparing 1,5-benzothiazepine derivatives of the formula wherein Ar is a phenyl substituted with a lower alkoxy, R is a lower alkyl, R 1 and R 2 are each a lower alkyl, and Y is a lower alkylene, which have excellent coronary vasodilating and psychoneurotic activities and are useful particularly as a Ca ++ -antagonistic coronary vasodilator.
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