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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-215
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-215
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filingDate 1982-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_52bb141b5edcb69fe338f373d8f5f7f6
publicationDate 1983-07-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0082873-A1
titleOfInvention COMPOSITIONS FOR TREATING GLAUCOMA.
abstract Method for treating glaucoma or lowering intraocular pressure in a mammal, and comprising administering locally to the eye of this mammal a selectively metabolized beta-blocking compound of formula: $ (6,) $ where R can be an alkyl lower, lower alkynyl, aryl, or aralkyl; A may be a direct bond, lower alkylenyl, or lower alkenyl; x can be an integer from 1 to 3; Ar can be a substituted or unsubstituted aromatic group; R1 can be lower alkyl, hydroxy lower alkyl, lower alkenyl, lower alkynyl, or aralkyl; and their pharmaceutically acceptable salts. Because of the relatively long duration of the effect of these compounds on ocular fluids and the relatively short duration of their effect on the systemic circulation, these compounds are useful for the treatment of excessive intraocular pressure without it occurring sensitive systemic side effects.
priorityDate 1981-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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