http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EA-034525-B1

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filingDate 2015-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1375d748c268f74fd458647c5c0fd655
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7d58514bb3a4df483ddcd4b990988f8a
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publicationDate 2020-02-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EA-034525-B1
titleOfInvention 2-Aryl-4-hydroxy-1,3-thiazole derivatives for use as TRPM8 inhibitors in the treatment of neuralgia, pain, chronic obstructive pulmonary disease and asthma
abstract The invention relates to compounds acting as selective antagonists of 8 members of the subfamily M of the cation channel of the transient receptor potential (TRPM8) and having the formula (I) These compounds are used in the treatment of diseases associated with TRPM8 activity, such as pain, inflammation, ischemia, neurodegeneration, stroke, mental disorders, pruritus, irritable bowel diseases caused by colds and / or exacerbated respiratory disorders and urological disorders.
priorityDate 2014-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 395.