| Predicate |
Object |
| assignee |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_50eb752940fa4aa36756a6bc9f6f3504 |
| classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-421
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-5365
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D498-18
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D263-46 |
| classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D498-18
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D263-46 |
| filingDate |
2016-03-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_02fcb4341a9f93ce1ad20809194ce2c5
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b456d0dc1f5de50e0c7a02bc4b24aa67
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_51bc59fbacab828cea740a0d3dada095
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e6c514632674c8e2ef2092f745709fac |
| publicationDate |
2019-11-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber |
EA-032630-B9 |
| titleOfInvention |
Amino Acid Acylation Reagents and Methods for Their Use |
| abstract |
The proposed compound of formula (I) or its salt, where R and R each are methyl; a compound of formula (Iaa) wherein the compound is stereoisomerically pure; as well as a method for producing a compound of formula (II) comprising contacting a compound of formula (I) with a nucleophile in the presence of one or more Lewis acids and one or more bases; a process for preparing a compound of formula (I) or a salt thereof, wherein R and R each are methyl, which comprises contacting a compound of formula (III) with 1,1'-thiocarbonyldiimidazole in the presence of one or more bases. |
| priorityDate |
2015-03-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type |
http://data.epo.org/linked-data/def/patent/Publication |