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publicationDate 2019-04-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EA-032124-B1
titleOfInvention ARILETHER AND THEIR APPLICATION
abstract The present invention relates to inhibitors of HIF-2α and to methods for their preparation and use for the treatment of malignant tumors. Certain compounds were active in a HIF-2α scintillation assay, a luciferase assay and VEGF ELISA assay, and resulted in a reduction in the size and regression of tumors in in vivo 786-O mice.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415791935
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419576099
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420235675
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID117942353
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419521000
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5324184
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449360014
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID117942143
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID547667
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID117942347
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID375056
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122506316
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6H8T0

Total number of triples: 1245.