abstract |
The present invention relates to a cyclosporin emulsion comprising: i) cyclosporin, ii) natural oil (long chain triglyceride), iii) phosphatidylcholine, iv) glycerin, v) pharmaceutically acceptable alkaline salt of free fatty acid, vi) oil containing medium chain triglycerides, vii) if necessary, hydrochloric acid or sodium hydroxide to adjust pH, viii) water. |