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filingDate 2013-01-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1280f61da7787bb8ff16fd75ba8906f9
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_88cc738d1df7a0dec4c159f558c286a7
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publicationDate 2017-06-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EA-027059-B1
titleOfInvention Fluoromethyl-5,6-dihydro-4H- [1,3] oxazines
abstract The present invention provides compounds of formula Ia-1 possessing β-secretase 1 inhibitor (BACE1) activity, preparation thereof, pharmaceutical compositions containing such compounds, and their use as therapeutically active substances for treating and / or preventing diseases and disorders characterized by an elevated β level. α-amyloid, and / or β-amyloid oligomers, and / or β-amyloid plaques and other deposits, such as Alzheimer's disease.
priorityDate 2012-01-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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