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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-12
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filingDate 2013-06-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_61b7fd4bbec84335debed33adb09590f
publicationDate 2016-12-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EA-025273-B1
titleOfInvention DIFTORGEXAHYDROCYCLOPENTAXOXASYNYLES AND DIFTORGEXAHYDROBENZOXASYNYLES AS BETA SECRETASE INHIBITORS
abstract The present invention proposed difluoro-cyclopentaoxazinyls and difluoro-benzooxazinyls of formula I, which have inhibitory activity against beta-secretase 1 (BACE1 from the English "beta-secretase 1"), their preparation, pharmaceutical compositions containing them and their use as therapeutically active substances. The active compounds of the present invention are useful in therapeutic and / or prophylactic treatment, for example, Alzheimer's disease.
priorityDate 2012-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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