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filingDate 2011-02-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2014-11-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EA-020528-B1
titleOfInvention MACRO CYCLES AS INHIBITORS OF XIA FACTOR
abstract The present invention relates to compounds of formula (I) or their stereoisomer, tautomer or pharmaceutically acceptable salt, where all variables are defined in the description of the invention. These compounds are selective factor XIa inhibitors or dual-action inhibitors of factor XIa and plasma kallikrein and can be used to treat thromboembolic and / or inflammatory disorders.
priorityDate 2010-02-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419494133
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GKA1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06880
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2155
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19221
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60947
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47776
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID177
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID931
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419541365
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100006947
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID43736
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68153
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393769
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24232
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415914366
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410011433
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453567348
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID185000
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID102122446
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16621
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID463117
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67930
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419525472
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426185522
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136415251
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A5F4BTH8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID459296
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426264250
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2734669
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16644
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47851
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID82189
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20391
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410605189
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00734
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID619414
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457465597
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08697
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419547992
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408912300
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67931
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410605182
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID140575537
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID19831830
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424322231
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419536034
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281407
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453757922
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403838
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424322216
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419558919
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID83172
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20392
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2736304
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID21788
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396985
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID617960
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100125764
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID565329
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424384073
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54687
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416163361
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450418934
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO13306
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23349072
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424355673
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393652
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID282522
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP87391
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452148691
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12299
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449111295

Total number of triples: 1344.