http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EA-020128-B1

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filingDate 2010-12-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5ef2565f4c15ba99d82d28efe6ecf8d3
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publicationDate 2014-08-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EA-020128-B1
titleOfInvention INHIBITORS DIACILGLYCEROLACILTRANSFERASE AND PHARMACEUTICAL COMPOSITION INCLUDING THEM
abstract The invention relates to a compound of formula (I) or a pharmaceutically acceptable salt thereof, wherein R is selected from the group consisting of H, F, Cl, —CF, —CH, —OH, —O (C-C1-6 alkyl), —O-cyclopropyl, O-CH-phenyl, —OC (H) F, and —OCF, R is selected from the group consisting of H and —CH, R is selected from the group consisting of H and —CH, provided that at least one of the group consisting of R and R represents H, and n is 1, 2 or 3, as diacylglycerol acyl transferase 1 (DGAT-1) inhibitors. The present invention also relates to a pharmaceutical composition containing the compound, and to the use of the compound as a medicament for the treatment of diabetes and / or obesity.
priorityDate 2009-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413715223
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A651
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1KJU9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419996541
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13190
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKA8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11723
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO75907
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420005425
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID521998
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4V9F0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKA5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424869160
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413714813
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKA6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70374856
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419985199
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419484328
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41522
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKA3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01342
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415956136

Total number of triples: 325.