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filingDate 2003-01-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c896dd2306666c0c8fd449bb7c12c45d
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publicationDate 2006-12-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EA-007738-B1
titleOfInvention MACROCYCLIC PEPTIDES WITH ACTIVITY AGAINST THE HEPATITIS C VIRUS
abstract The compounds of formula (I) in which R is hydroxy or NHSOR, where R is C-C1-6alkyl, C-Cycloalkyl or C-C1-6alkyl-C-Cycloalkyl, which are all optionally substituted with 1 to 3 substituents selected from the group consisting of halogen, cyano, nitro, OS-C1-6alkyl, amido, amino or phenyl, or R is C- or Saryl, optionally substituted with 1-3 substituents selected from the group consisting of halogen, cyano, nitro, C-C1-6alkyl, OS-C1-6alkyl, amido, amino or phenyl; R is C-Cycloalkyl and R is cyclopentyl; or their pharmaceutically acceptable salts, which can be used as inhibitors of the NS3 protease HCV.
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type http://data.epo.org/linked-data/def/patent/Publication

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