http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EA-004512-B1
Outgoing Links
Predicate | Object |
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assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_a717ea5b2ac78ac329ab3a9659d834d2 http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_a4b14e936224599e9ceef6151c235adf |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D265-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-10 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F9-6533 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D265-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D265-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P15-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-537 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-536 |
filingDate | 2000-05-01-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bf79bece1af25e46716dd60ac601d773 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8ebb5d80c95bd67b245de851fdd64050 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b6f18a51ba775a6a9666cfac348cb060 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ef0217e26f854b6936c258047b15d014 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_588e65de7f4150013e2a9f3227a9282c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_22de4bd174d72fd1cecf8456ec5f6609 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0569843abdd8c901960ac3299f5290af http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_535d7c9a1f0b479f89c976b799c73ec8 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d33b37b7d3e2705a02f4d2b2007fcfd6 |
publicationDate | 2004-04-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | EA-004512-B1 |
titleOfInvention | CYCLOCARBAMATE DERIVATIVES AS PROTESTERONE RECEPTOR MODULATORS |
abstract | The invention relates to compounds of the formula where R and R are independent substituents selected from the group consisting of H, C -C alkyl, substituted C-C alkyl, C-C alkenyl, substituted C-C alkenyl, C-C alkynyl, substituted C-C alkynyl, C-C cycloalkyl, substituted C-C cycloalkyl, aryl, substituted aryl, heterocyclyl, substituted heterocyclyl COR, or NRCOR; or R and R are fused to form a saturated or unsaturated 3-8 membered spirocyclic ring optionally containing in its skeleton from one to three heteroatoms selected from the group consisting of O, S and N; wherein the ring may be optionally substituted with 1-4 substituents selected from the group consisting of fluoro, C -C alkyl, C -C alkoxy, C -C thioalkyl, CF, OH, CN, NH, NH (C -C alkyl) or N (C -C alkyl) ); R 2 is selected from H, C -C alkyl, substituted C -C alkyl, aryl, substituted aryl, C -C alkoxy, substituted C -C alkoxy, C -C aminoalkyl, or substituted C -C aminoalkyl; R5 is H, C -C alkyl, or substituted C -C alkyl; R5 is H, OH, NH, C -C alkyl, substituted C -C alkyl, C -C alkenyl, substituted C -C alkenyl, alkynyl, substituted alkynyl, or COR; R5 is H, C -C alkyl, substituted C -C alkyl, aryl, substituted aryl, C -C alkoxy, substituted C -C alkoxy, C -C aminoalkyl, or substituted C -C aminoalkyl; R5 is H, halogen, CN, NO, C -C alkyl, substituted C -C alkyl, alkynyl, substituted alkynyl, C -C alkoxy, substituted C -C alkoxy, amino, C -C aminoalkyl, or substituted C -C aminoalkyl; R is selected from the group consisting of a substituted benzene ring containing substituents X, Y and Z as defined in the claims, or a five or six membered ring with 1,2 or 3 heteroatoms in the ring selected from the group consisting of O, S, SO, SO, or NR containing one or two independent substituents defined in the claims; R is absent or is H, O, |
priorityDate | 1999-05-04-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
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