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filingDate 2000-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2004-06-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_721f42fe50043b4e4f714c345c5deef6
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0f7d05a1a8341ad6fabd098f6c34e37f
publicationDate 2004-06-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber DE-60005017-T2
titleOfInvention PRODRUGS OF IMPDH INHIBITING CARBAMATES
abstract The present invention relates to novel compounds, methods of preparing these compounds, and pharmaceutical compositions comprising these compounds. These compounds are carbamate prodrugs that convert to active inhibitors of the IMPDH enzyme in vivo. The compounds and pharmaceutical compositions of this invention are particularly well suited for activation and subsequent inhibition of the IMPDH enzyme activity. Consequently, these prodrugs may be advantageously used as therapeutic agents for IMPDH mediated processes. This invention also relates to methods for inhibiting the activity of IMPDH using the compounds and compositions of this invention.
priorityDate 1999-06-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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