http://rdf.ncbi.nlm.nih.gov/pubchem/patent/DE-2457971-A1
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_eccd894c99fea2d1c0c8735872bb2309 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 |
filingDate | 1974-12-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6e916f31639371f6e47e94ef219e8e50 |
publicationDate | 1976-06-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | DE-2457971-A1 |
titleOfInvention | PROCESS FOR THE PREPARATION OF 2-ACYL4-OXO-PYRAZINO-ISOCHINOLINE DERIVATIVES |
abstract | Compounds of the formula I <IMAGE> in which -CO-R denotes an acyl radical of a carboxylic acid, in which the radical R denotes hydrogen or contains up to 25 C atoms are prepared by cyclisation under HE-eliminating conditions of a compound of the formula II <IMAGE> in which E denotes OH, alkylsulphonyloxy having 1-6 C atoms, arylsulphonyloxy having 6-10 C atoms, acyloxy having 1-7 C atoms, the acyl radical being derived from a carboxylic acid, tetrahydropyranyl-2-oxy, alkoxy having 1-4 C atoms, Cl, Br or I. The compounds have outstanding parasitological and pharmacological properties together with good tolerability. They act, inter alia, as useful anthelmintics and in particular display a broad spectrum of action against cestodes and trematodes. Psychotropic properties and properties affecting blood pressure can also occur. |
isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-4195984-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0086678-A1 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-4497952-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/FR-2533925-A1 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-4217452-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-4254031-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/FR-2520740-A1 |
priorityDate | 1974-12-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 147.