http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CZ-9904752-A3

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_f00b503b4045fc858275a7c77e27c087
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-20
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P29-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-20
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-445
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-505
filingDate 1998-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fc921db55ff811629a5cf328e7da323f
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a11bece7929dd45b4d937d515918d004
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e437aa3d64c0042007aa13759d38fa6f
publicationDate 2000-10-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CZ-9904752-A3
titleOfInvention Aminospivopiperidinequinazoline Derivatives
abstract The present invention provides compounds of formula (I), venwherein A represents an aromatic carbocyclic ring or a five or fivena six membered heterocyclic aromatic ring containing 1nup to 3 heteroatoms which may be the same or different and arenselected from oxygen, nitrogen and sulfur; X represents a groupnof formula - (CH 2) n -, wherein n is zero or 1; and R 1, R 2 and R 3nare defined in the specification and their pharmaceutically acceptable saltsnand their enantiomers and tautomers; together with theirsnpreparations, preparations containing them and their use in therapy.nThe compounds are nitric oxide synthase inhibitors and hencenthey are particularly suitable for the treatment or prophylaxis of inflammatory diseasesndiseases and boles
priorityDate 1998-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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