http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CZ-280603-B6
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_05a203d85ee01909eaf728dc16f0f6cb |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-47 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-08 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-233 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D519-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-435 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P31-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-47 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4738 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4375 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-08 |
| filingDate | 1993-04-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_54a2dbaf3e0767d2c6b8dced6ebca561 |
| publicationDate | 1996-03-13-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | CZ-280603-B6 |
| titleOfInvention | Quinoline and naphryridine derivatives and antibacterial agents based thereon |
| abstract | The quinoline and naphthyridine derivatives of formula I wherein A is CH, CF or N; Y represents ethyl, cyclopropyl, 4-fluorophenyl or 2,4-difluorophenyl; or A and Y taken together represent O-CH.sub.2.n.-CH (CH.sub.3.n.) - C, CH.sub.2.n.-CH.sub.2.n. -CH (CH 3) - C or O-CH (CH 3) - NC; R.sub.1.n. represents hydrogen or methyl; and R.sub.2.n. represents hydrogen, 5-methyl-2,5-diazabicyclo [2.2.1] hept-2-yl, 8-methyl-3,8-diazabicyclo [3.2.2] non-4-yl; wherein if R.sub.2.n. represents a hydrogen atom, then A and Y together represent a group of the formula CH.sub.2.n.-CH.sub.2.n.-CH (CH.sub.3.n.) -C; and pharmaceutically acceptable acid addition salts thereof, provided that R.sub.2.n. is different from hydrogen. The invention further relates to an antibacterial composition based thereon. These derivatives, which contain a 3-carboxaldehyde group, are prodrugs which can be used for the treatment of bacterial infections, in particular in the form of injectables. As a specific example |
| priorityDate | 1992-07-15-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
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