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filingDate 2001-08-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e1e9078a30d1e5c0ccf05ea611776a71
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_34af450328dd7d686e4081d0dab88740
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publicationDate 2003-08-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CZ-2003414-A3
titleOfInvention Azaamino acid derivatives as Factor Xa inhibitors 15, a process for their preparation, intermediates for this preparation, their use, and a pharmaceutical composition containing them
abstract The invention relates to semicarbicides of the general formula (I), wherein R<1>, R<2>, R<3>, R<4> and I are defined as in claim 1. The compounds of formula (I) can be used as active ingredients for medicaments in human and veterinary medicine, especially for combating and preventing thromboembolic diseases such as thrombosis, myocardial infarction, arteriosclerosis, inflammations, apoplexy, angina pectoris, restenosis after angioplasty, intermittent claudication, tumors, tumor diseases and/or tumor metastases.
priorityDate 2000-08-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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